Structure determination and comparison of BM567, a sulfonylurea, with terbogrel, two compounds with dual action, thromboxane receptor antagonism and thromboxane synthase inhibition

Catherine Michaux; Stéphanie Rolin; Jean-Michel Dogne; François Durant; Bernard Masereel; Jacques Delarge; Johan Wouters

doi:10.1016/S0960-894X(01)00114-7

Structure determination and comparison of BM567, a sulfonylurea, with terbogrel, two compounds with dual action, thromboxane receptor antagonism and thromboxane synthase inhibition

Catherine Michaux, Stéphanie Rolin, Jean-Michel Dogne, François Durant, Bernard Masereel, Jacques Delarge, Johan Wouters

Unite de recherche en chimie physique, theorique et structurale

Résultats de recherche: Contribution à un journal/une revue › Article › Revue par des pairs

Résumé

BM567, a sulfonylurea compound - whose crystal structure is here discussed - and terbogrel, are both thromboxane receptor antagonists and thromboxane synthase inhibitors. In this paper, their crystallographic and electronic structures are compared and lead to new synthesis prospects among the sulfonylurea series.

langue originale	Anglais
Pages (de - à)	1019-1022
Nombre de pages	4
journal	Bioorganic & Medicinal Chemistry Letters
Volume	11
Numéro de publication	8
Les DOIs	https://doi.org/10.1016/S0960-894X(01)00114-7
Etat de la publication	Publié - 23 avr. 2001

Accès au document

10.1016/S0960-894X(01)00114-7

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Contient cette citation

Michaux, C., Rolin, S., Dogne, J.-M., Durant, F., Masereel, B., Delarge, J., & Wouters, J. (2001). Structure determination and comparison of BM567, a sulfonylurea, with terbogrel, two compounds with dual action, thromboxane receptor antagonism and thromboxane synthase inhibition. Bioorganic & Medicinal Chemistry Letters, 11(8), 1019-1022. https://doi.org/10.1016/S0960-894X(01)00114-7

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title = "Structure determination and comparison of BM567, a sulfonylurea, with terbogrel, two compounds with dual action, thromboxane receptor antagonism and thromboxane synthase inhibition",

abstract = "BM567, a sulfonylurea compound - whose crystal structure is here discussed - and terbogrel, are both thromboxane receptor antagonists and thromboxane synthase inhibitors. In this paper, their crystallographic and electronic structures are compared and lead to new synthesis prospects among the sulfonylurea series.",

author = "Catherine Michaux and St{\'e}phanie Rolin and Jean-Michel Dogne and Fran{\c c}ois Durant and Bernard Masereel and Jacques Delarge and Johan Wouters",

year = "2001",

month = apr,

day = "23",

doi = "10.1016/S0960-894X(01)00114-7",

language = "English",

volume = "11",

pages = "1019--1022",

journal = "Bioorganic & Medicinal Chemistry Letters",

issn = "0960-894X",

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number = "8",

}

Michaux, C, Rolin, S, Dogne, J-M , Durant, F , Masereel, B, Delarge, J & Wouters, J 2001, 'Structure determination and comparison of BM567, a sulfonylurea, with terbogrel, two compounds with dual action, thromboxane receptor antagonism and thromboxane synthase inhibition', Bioorganic & Medicinal Chemistry Letters, VOL. 11, Numéro 8, p. 1019-1022. https://doi.org/10.1016/S0960-894X(01)00114-7

Structure determination and comparison of BM567, a sulfonylurea, with terbogrel, two compounds with dual action, thromboxane receptor antagonism and thromboxane synthase inhibition. / Michaux, Catherine; Rolin, Stéphanie; Dogne, Jean-Michel et al.
Dans: Bioorganic & Medicinal Chemistry Letters, Vol 11, Numéro 8, 23.04.2001, p. 1019-1022.

Résultats de recherche: Contribution à un journal/une revue › Article › Revue par des pairs

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AU - Michaux, Catherine

AU - Rolin, Stéphanie

AU - Dogne, Jean-Michel

AU - Durant, François

AU - Masereel, Bernard

AU - Delarge, Jacques

AU - Wouters, Johan

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AB - BM567, a sulfonylurea compound - whose crystal structure is here discussed - and terbogrel, are both thromboxane receptor antagonists and thromboxane synthase inhibitors. In this paper, their crystallographic and electronic structures are compared and lead to new synthesis prospects among the sulfonylurea series.

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