University of Namur

  • Belgium

Research Output

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Literature review
1989

New torasemide derivatives inhibit brain slices and astrocytes swelling induced by potassium

Masereel, B., Grisar, T., Delarge, J. & Burette, M., 1989, In : Journal of Neurochemistry. 52, p. S183

Research output: Contribution to journalLiterature review

1990

New lipophilic torasemide derivatives inhibit astrocytic potassium uptake and rat brain slices water uptake

Masereel, B., Schynts, M. & Delarge, J., 1990, In : Journal de Pharmacie de Belgique. 45, (1)

Research output: Contribution to journalLiterature review

New sulfonylurea derivatives as potential antihypertensive drugs

Masereel, B., Pirotte, B., Schynts, M., Ferrari, P., Thunus, L. & Delarge, J., 1990, In : Journal de Pharmacie de Belgique. 45, p. 405

Research output: Contribution to journalLiterature review

Structure-activity of sulfonylurea compounds (SUC) on Na-Cl transport in isolated perfused rabbit cortical thick ascending limbs of Henle's loop

Lohrmann, E., Nitschke, R., Schlatter, E., Masereel, B., Delarge, J., Lang, HJ., Englert, HC. & Greger, R., 1990, In : European Journal of Physiology. 415, suppl 1, p. R40

Research output: Contribution to journalLiterature review

Structure-activity relationship of new torasemide derivatives on Na-K-2Cl cotransporter in perfused rabbit thick ascending limb of Henle's loop

Masereel, B., Pirotte, B., Schynts, M., Delarge, J., Lohrmann, E., Nitschke, R., Schlatter, E. & Greger, R., 1990, In : Pharmaceutisch Weekblad. 12, p. E7

Research output: Contribution to journalLiterature review

1991

4-Amino-4H-1,2,4-triazole and 5-aminothiazole derivatives structurally related to ß -lactam antibiotics as potential inhibitors of serine proteases

Boggetto, N., Vilain, A. C., Pirotte, B., Masereel, B., Vergely, I., Dupont, L., Delarge, J. & Reboud, M., 1991, In : Archieve der Pharmazie. 324, p. 658

Research output: Contribution to journalLiterature review

Inhibiteurs potentiels de protéases à sérine apparentés aux antibiotiques ß-lactamiques

Pirotte, B., Vilain, A. C., Vergely, I., Boggetto, N., Masereel, B., Dupont, L., Delarge, J. & Reboud, M., 1991, In : Regard sur la Biochimie. 6, p. 91

Research output: Contribution to journalLiterature review

Loop diuretics: SAR, molecular interactions and target topography

Masereel, B., Dupont, L., Lohrmann, E., Schynts, M., Pirotte, B., Greger, R. & Delarge, J., 1991, In : Archieve der Pharmazie. 324, p. 650

Research output: Contribution to journalLiterature review

1992

3-Oxo-2H,4H-pyrido [2,3-e] [1,2,4]-thiadiazine 1,1-dioxide, a sweetening agent of the sulfonamide family structurally related to saccharin and acesulfame

Pirotte, B., de Tullio, P., Masereel, B., Parmentier, M., Schynts, M. & Delarge, J., 1992, In : Pharmaceutische Weekblad. 14, suppl, p. I10

Research output: Contribution to journalLiterature review

New dihydrocoumarin derivatives as potential mechanism-based inactivators of serine proteinases

Schynts, M., Boggetto, N., Masereel, B., Pirotte, B., Fesquet, S., Vergely, I., Delarge, J. & Reboud, M., 1992, In : Pharmaceutische Weekblad. 14, suppl, p. I11

Research output: Contribution to journalLiterature review

New relative K+-sparing high ceiling diuretics related to torasemide

Masereel, B., Schynts, M., Lohrmann, E., Pirotte, B., Greger, R. & Delarge, J., 1992, In : Journal de Pharmacie de Belgique. 47, p. 447

Research output: Contribution to journalLiterature review

1993

Improved pancreatic K-ATP channel openers belonging to the pyridothiadiazine chemical class

Pirotte, B., de Tullio, P., Lebrun, P., Antoine, M-H., Masereel, B., Schynts, M. & Delarge, J., 1993, In : Journal de Pharmacie de Belgique. 48, (2), p. 143

Research output: Contribution to journalLiterature review

Loop diuretics and the renal Na+ K+ 2Cl- cotransport: Interaction model

Masereel, B., Schynts, M., Pirotte, B. & Delarge, J., 1993, In : Journal de Pharmacie de Belgique. 48, (2), p. 141

Research output: Contribution to journalLiterature review

1994

A novel coumarinic inhibitor inactivates cathepsin G but not human leukocyte elastase

Fesquet, S., Schynts, M., Boggetto, N., Masereel, B., Pirotte, B., Delarge, J., Jiang, KY. & Reboud, M., 1994, In : Journal de Pharmacie de Belgique. 49, (2), p. 258

Research output: Contribution to journalLiterature review

Etude structurale comparative du pinacidil, du diazoxide et du cromakalim, ouvreurs de canaux potassiques appartenant à trois classes chimiques distinctes

Dupont, L., Pirotte, B., de Tullio, P., Masereel, B., Schynts, M. & Delarge, J., 1994, In : Journal de Pharmacie de Belgique. 49, (2), p. 282

Research output: Contribution to journalLiterature review

Pharmacology of a new sulphonylurea (BM 27) effective in brain edema

Masereel, B., Schynts, M., Pirotte, B., de Tullio, P. & Delarge, J., 1994, In : Journal de Pharmacie de Belgique. 49, (1), p. 88

Research output: Contribution to journalLiterature review

Synthèse de dérivés 3-aminoaralkyl-2aryl-4H-pyrido [4,3-e]-1,2,4-thiadiazine 1,1-dioxydes et leur évaluation en tant qu'antagonistes de la cholécystokinine

de Tullio, P., Pirotte, B., Masereel, B., Diouf, O., Caignard, D. H., Renard, P. & Delarge, J., 1994, In : Journal de Pharmacie de Belgique. 49, (2), p. 244

Research output: Contribution to journalLiterature review

Synthesis of a series of 4H-1,2,4,-pyridothiadiazine 1,1-dioxydes and their evaluation as new potassium channel openers

de Tullio, P., Pirotte, B., Dupont, L., Lebrun, P., Antoine, M-H., Fontaine, J., Masereel, B., Schynts, M. & Delarge, J., 1994, In : Journal de Pharmacie de Belgique. 49, (1), p. 85

Research output: Contribution to journalLiterature review

1995

3-Arylcarboxamidomethyl-4H-pyrido [4,3-e]-1,2-4-thiadiazine 1,1-dioxydes en tant qu'antagonistes non-peptidiques de la cholécystokinine: synthèse et évaluation pharmacologique

Pirotte, B., de Tullio, P., Podona, T., Masereel, B., Caignard, D. H., Renard, P. & Delarge, J., 1995, In : Journal de Pharmacie de Belgique. 50, p. 253

Research output: Contribution to journalLiterature review

Synthesis and pharmacology of N"-(4-arylaminopyrid-3-yl)sulfonyl-N-cyano-N'-isopropylguanidines

Masereel, B., Schynts, M., Pirotte, B., de Tullio, P. & Delarge, J., 1995, In : Journal de Pharmacie de Belgique. 50, p. 250

Research output: Contribution to journalLiterature review

1996

2-,3- and 4-substituted pyrido[4,3-e]-1,2,4-thiadiazine 1,1-dioxides as ATP-sensitive potassium channel openers

de Tullio, P., Pirotte, B., Ouedraogo, R., Dupont, L., Lebrun, P., Fang, ZY., Masereel, B., Fontaine, J., Antoine, M-H., Neven, P., Pochet, L. & Delarge, J., 1996, In : Journal de Pharmacie de Belgique. 51, (1), p. 108

Research output: Contribution to journalLiterature review

3-Alkylamino-4H-pyrido[2,3-e]-1,2,4-thiadiazine 1,1-dioxides structurally related to both diazoxide and pinacidil: a new class of potassium channel openers

Pirotte, B., Khelili, S., de Tullio, P., Fang, ZY., Ouedraogo, R., Antoine, M-H., Fontaine, J., Masereel, B., Dewalque, D., Damas, J., Pochet, L., Delarge, J. & Lebrun, P., 1996, In : Journal de Pharmacie de Belgique. 51, (1), p. 117

Research output: Contribution to journalLiterature review

Anticonvulsant properties of 4-cycloalkyamino-pyrid-3-yl sulfonylureas and -thioureas

Masereel, B., Lambert, D., Bia, F., Diouf, O., Liégeois, J-F., de Tullio, P., Pirotte, B., Pochet, L., Khelili, S. & Delarge, J., 1996, In : Journal de Pharmacie de Belgique. 51, 3b, p. 17

Research output: Contribution to journalLiterature review

Attempts to stimulate thyroid tissues in vitro.

Bister, J-L., Derycke, G., Vandermeir, M-A. & Paquay, R., 1996, In : Eur. J. Physiol. . 431, R325

Research output: Contribution to journalLiterature review

Design and synthesis of aromatic esters and amides of 6-chloromethyl-2-oxo-2H-benzopyran-3 carboxylic acid as inhibitors of alpha-chymotrypsin

Pochet, L., Doucet, C., Schynts, M., Thierry, N., Boggetto, N., Pirotte, B., Masereel, B., de Tullio, P., Delarge, J. & Reboud-Ravaux, M., 1996, In : Journal de Pharmacie de Belgique. 51, (1), p. 117

Research output: Contribution to journalLiterature review

Les canaux potassiques ATP-dépendants et la secrétion d'insuline. Effets du BPDZ 62

Ouedraogo, R., Pirotte, B., Antoine, M-H., de Tullio, P., Masereel, B., Dunne, M., Kane, C. & Lebrun, P., 1996, In : Journal de Pharmacie de Belgique. 51, 3b, p. 41

Research output: Contribution to journalLiterature review

Nouveaux dérivés de l'acide 6-chloromé thyl-2-oxo-2H-1-benzopyran-3-carboxylique en tant qu' inhibiteurs de protéases à sérine: étude des relations structure-activité explicant leur sélectivité d'action

Doucet, C., Pochet, L., Schynts, M., Pirotte, B., Thierry, N., Boggetto, N., Masereel, B., de Tullio, P., Delarge, J. & Reboud-Ravaux, M., 1996, In : Journal de Pharmacie de Belgique. 51, 3b, p. 18

Research output: Contribution to journalLiterature review

Nouvelles stratégies de synthèse des pyridothiadiazinedioxydes structuralement apparentées au diazoxide

Khelili, S., Pirotte, B., de Tullio, P., Masereel, B. & Delarge, J., 1996, In : Journal de Pharmacie de Belgique. 51, 3b, p. 19

Research output: Contribution to journalLiterature review

Synthèse de nouvelles pyridothiadiazines et leur évaluation en tant que modulateurs des récepteurs glutamatergiques à l'acide alpha-amino-3-hydroxy-5-méthyl-4-isoxazolepropionique

Diouf, O., Pirotte, B., Podona, T., de Tullio, P., Masereel, B., Delarge, J., Morain, P. & Lepagnol, J., 1996, In : Journal de Pharmacie de Belgique. 51, 3b, p. 20

Research output: Contribution to journalLiterature review

Synthesis, bioavailability and anticonvulsant activity of 2-cyanoguanidinophenytoin, a structural analogue of phenytoin

Lambert, D., Masereel, B., Gallez, D., Geurts, M. & Scriba, G., 1996, In : Journal de Pharmacie de Belgique. 51, (1), p. 113

Research output: Contribution to journalLiterature review

The selectivity of some pyridobenzazepine derivatives for the dopamine D4 receptor

Liégeois, J-F., Bruhwyler, J., Damas, J., Rogister, F., Masereel, B., Geczy, J. & Delarge, J., 1996, In : Journal de Pharmacie de Belgique. 51, 3b, p. 16

Research output: Contribution to journalLiterature review

1998

Insulinotropic effect of glibenclamide isosteres

Nguyen, Q. A., Pochet, L., Ouedraogo, R., Dunne, M. J., Masereel, B., Lebrun, P. & Antoine, M-H., 1998, In : Fundamental and Clinical Pharmacology. 12, p. 307

Research output: Contribution to journalLiterature review

Ovarian activity and fertilisation possibilities in local Burundian ewes and goats.

Mbayahaga, J. N., 1998, In : Journal of Reproduction and Fertility. 19, Abs 65

Research output: Contribution to journalLiterature review

R. STRAUB, David Aubert, "escripvain" et "clerc", Amsterdam-Atlanta, Rodopi, 1995

Palumbo, G. B., 1998, In : Medioevo Romanzo. XXII, p. 156-157 2 p.

Research output: Contribution to journalLiterature review

Waltharius: Epica e Saga da Virgilio ai 'Nibelunghi', a cura di E. D'ANGELO, Milano-Trento, Luni, 1998

Palumbo, G. B., 1998, In : Medioevo Romanzo. XXII, p. 454-455 2 p.

Research output: Contribution to journalLiterature review

1999

Antiplatelet properties of BM-519, a novel combined thromboxane A2 receptor antagonist and thromboxane synthase inhibitor

Dogné, J-M., de Leval, X., Delarge, J., Neven, P., Rolin, S., David, J-L., Fillet, G. & Masereel, B., 1999, In : Blood. 94, (suppl 1), p. 3625

Research output: Contribution to journalLiterature review

BM-519, a novel non-carboxylic thromboxane A2 antagonist

Masereel, B., Lacan, F., Fontaine, J., Nuhrich, A., Delarge, J., Pochet, L. & Dogné, J-M., 1999, In : Fundamental and Clinical Pharmacology. 13, (suppl 1), p. 191s

Research output: Contribution to journalLiterature review

Hugues Ripelin de Strasbourg, Le Somme Abregiet de Theologie

Laoureux, S., 1999, In : Le Moyen Âge. 105, p. 861-864 4 p.

Research output: Contribution to journalLiterature review

In vivo and in vitro effect of new glibenclamides isosteres

Lebrun, P., Ouedraogo, R., Nguyen, QA., Antoine, M-H., Dunne, M. J., Pirotte, B. & Masereel, B., 1999, In : Fundamental and Clinical Pharmacology. 13, (suppl 1), p. 381s

Research output: Contribution to journalLiterature review

Maître Eckhart, L¿étincelle de l'âme

Laoureux, S., 1999, In : Le Moyen Âge. 105, p. 558-561 4 p.

Research output: Contribution to journalLiterature review

PFA-100, a novel pharmacological tool for characterization of antiplatelet potency of thromboxane receptor antagonists

Dogné, J-M., de Leval, X., Delarge, J., Neven, P., Rolin, S., David, J-L., Fillet, G. & Masereel, B., 1999, In : Blood. 94 (suppl 1), p. 3626

Research output: Contribution to journalLiterature review

2000

Characterization of the antiplatelet activity of ticlopidine and acetylsalicylic acid by PFA-100

Dogné, J-M., de Leval, X., Neven, P., Rolin, S., David, J-L., Delarge, J. & Masereel, B., 2000, In : Fundamental and Clinical Pharmacology. 14, p. 168

Research output: Contribution to journalLiterature review

Design, synthesis and pharmacological evalution of original thromboxane receptor antagonists.

Dogné, J-M., de Leval, X., Delarge, J., Reginster, J-Y., Henrottin, Y., Neven, P., Rolin, S. & Masereel, B., 2000, In : Mediators of Inflammation. 9, p. 53

Research output: Contribution to journalLiterature review

Design and pharmacological evaluation of a novel combined thromboxane A2 receptor antagonist and thromboxane synthase inhibitor derived from torasemide as promising antiplatelet agent

Dogné, J-M., de Leval, X., Rolin, S., Neven, P., Kolh, P., David, J-L., Fillet, G., Delarge, J. & Masereel, B., 2000, In : Blood. 96, 11, p. 230

Research output: Contribution to journalLiterature review

Effects of TXA2 receptor antagonists derived from torasemide on platelet function

Dogné, J-M., de Leval, X., Neven, P., Rolin, S., Somers, F., David, J-L., Delarge, J. & Masereel, B., 2000, In : Fundamental and Clinical Pharmacology. 14, p. 168

Research output: Contribution to journalLiterature review

Evaluation of classical NSAIDs on COX-1 and COX-2 purified enzymes and prognosis of their effects on physiological responses

de Leval, X., Henrotin, Y., Masereel, B., Somers, F., Neven, P., Devel, P., Delarge, J. & Dogné, J-M., 2000, In : Fundamental and Clinical Pharmacology. 14, p. 167

Research output: Contribution to journalLiterature review

Inhibition of cellular invasion by 3-chlorophenyl 6-(acétoxymethyl)-2-oxo-2H-1-benzopyran-3-carboxylate

Kempen, I., Pochet, L., Papapostolu, D., Bogetto, N., Doucet, C., Masereel, B., Foidart, J-M., Reboud-Ravaux, M., Frankenne, F. & Pirotte, B., 2000, In : European Journal of Physiology. 440, (78), p. R252

Research output: Contribution to journalLiterature review