Résultat de recherche 2011 2017

  • 45 Citations
  • 3 h-Index
  • 5 Poster
  • 4 Article
  • 3 Article dans les actes d'une conférence/un colloque
2017

An optimized dRVVT-based assay to estimate the intensity of anticoagulation in patients treated with direct oral anticoagulants

Sennesael, A-L., Exner, T., Chatelain, B., Lessire, S., Larock, A-S., Vancraeynest, C., Pochet, L., Dogné, J-M., Spinewine, A., Mullier, F. & Douxfils, J. 2017 (Accepté/sous presse) Dans : Thrombosis Research.

Résultats de recherche: Recherche - Revue par des pairsArticle

Prothrombin Time
Anticoagulants
2015

3D-QSAR, design, synthesis and characterization of trisubstituted harmine derivatives with in vitro antiproliferative properties

Meinguet, C., Bruyère, C., Frédérick, R., Mathieu, V., Vancraeynest, C., Pochet, L., Laloy, J., Mortier, J., Wolber, G., Kiss, R., Masereel, B. & Wouters, J. 13 avr. 2015 Dans : European Journal of Medicinal Chemistry. 94, p. 45-55 11 p., 7726

Résultats de recherche: Recherche - Revue par des pairsArticle

Accès ouvert
Harmine
Quantitative Structure-Activity Relationship
Solubility
In Vitro Techniques
Derivatives
2014
Indoleamine-Pyrrole 2,3,-Dioxygenase
thiosemicarbazide
Derivatives
Scaffolds
Substitution reactions

Thiosemicarbazide Derivatives as Novel Indolamine-2,3-dioxygenase (IDO) Inhibitors

Serra, S., Moineaux, L., Vancraeynest, C., Masereel, B., Pochet, L., Wouters, J. & Frédérick, R. 2014 Chemmedchem EFMC-ISMC 2014 Book of Abstracts. p. 280

Résultats de recherche: RechercheArticle dans les actes d'une conférence/un colloque

2013

coauthor on lecture: NOVEL DEVELOPMENT IN COUMARINS AS FXIIa INHIBITORS: IMPROVEMENT OF SOLUBILITY

Bouckaert, C., Vancraeynest, C., Dolušić, E., Frédérick, R. & Pochet, L. 2013 Book of Abstracts, 27èmes Journées franco-belges de Pharmacochimie / 21èmes Conférences européennes du GP2A. Vol OC05

Résultats de recherche: RechercheArticle dans les actes d'une conférence/un colloque

Accès ouvert
!!File
Factor XIIa
Coumarins
Solubility
factor XIIa inhibitor
Hemorrhage

Design and synthesis of thiosemicarbazides as inhibitors of Arginase I, a therapeutic target for anticancer immunotherapy

Colette, C., Vancraeynest, C., Serra, S., Pochet, L. & Frédérick, R. 2013 2013 Book of Abstracts, 27èmes Journées franco-belges de Pharmacochimie / 21èmes Conférences européennes du GP2A. p. 45

Résultats de recherche: RechercheArticle dans les actes d'une conférence/un colloque

Accès ouvert
!!File
Coumarins
Solubility
factor XIIa inhibitor
Factor XIIa
Thrombosis
2012

Novel trisubstituted harmine derivatives with original in vitro anticancer activity

Frédérick, R., Bruyére, C., Vancraeynest, C., Reniers, J., Meinguet, C., Pochet, L., Backlund, A., Masereel, B., Kiss, R. & Wouters, J. 26 juil. 2012 Dans : Journal of medicinal chemistry. 55, 14, p. 6489-6501 13 p.

Résultats de recherche: Recherche - Revue par des pairsArticle

Harmine
Carbolines
Neoplasms
In Vitro Techniques
Growth

STUDY OF COUMARINS WITH IMPROVED SOLUBILITY TO INHIBIT FXIIa, AN EMERGING TARGET IN THROMBOSIS RESEARCH

Bouckaert, C., Vancraeynest, C., Dolušić, E., Frédérick, R. & Pochet, L. 30 nov. 2012 p. Book of Abstracts, MedChem 2012, Château de Colonster, Liège - November 30, 2012, P01 1 p.

Résultats de recherche: RecherchePoster

!!File
Factor XIIa
Coumarins
Solubility
Thrombosis
Research
2011

Aromatic Thiosemicarazones are inhibitors of tryptophan 2,3-Dioxygenase (TDO), an emerging target for cancer treatment

Dolusic, E., Modaffari, S., Larrieu, P., Vancraeynest, C., Pilotte, L., Colau, D., Stroobant, V., Wouters, J., Masereel, B., Van den Eynde, B. & Frédérick, R. 2011 p. Book of Abstracts, ASMC 11, St. Petersburg, Russia, August 21-25, 2011, P157 1 p.

Résultats de recherche: RecherchePoster

!!File
Tryptophan Oxygenase
Thiosemicarbazones
Oncology
Methisazone
Bearings (structural)

THIOSEMICARBAZONES AS INHIBITORS OF TRYPTOPHAN 2,3-DIOXYGENASE (TDO), AN EMERGING TARGET FOR CANCER TREATMENT

Dolusic, E., Modaffari, S., Larrieu, P., Vancraeynest, C., Pilotte, L., Colau, D., Stroobant, V., Van den Eynde, B., Wouters, J., Masereel, B. & Frédérick, R. 2011 p. Book of Abstracts, Annual One-Day Meeting on Medicinal Chemistry of SRC & KVCV (MedChem 2011), Ghent, 25 November 2011, p. 21 1 p.

Résultats de recherche: RecherchePoster

!!File
Tryptophan Oxygenase
Indoleamine-Pyrrole 2,3,-Dioxygenase
Thiosemicarbazones
Oncology
Enzymes