Résultat de recherche 2011 2017

  • 95 Citations
  • 6 h-Index
  • 8 Article
Filtre
Article
2017

A harmine-derived beta-carboline displays anti-cancer effects in vitro by targeting protein synthesis

Carvalho, A., Chu, J., Meinguet, C., Kiss, R., Vandenbussche, G., Masereel, B., Wouters, J., Kornienko, A., Pelletier, J. & Mathieu, V. 15 juin 2017 Dans : European Journal of Pharmacology. 805, p. 25-35 11 p.

Résultats de recherche: Contribution à un journal/une revueArticle

norharman
Harmine
Protein Transport
Neoplasms
In Vitro Techniques
2015

3D-QSAR, design, synthesis and characterization of trisubstituted harmine derivatives with in vitro antiproliferative properties

Meinguet, C., Bruyère, C., Frédérick, R., Mathieu, V., Vancraeynest, C., Pochet, L., Laloy, J., Mortier, J., Wolber, G., Kiss, R., Masereel, B. & Wouters, J. 13 avr. 2015 Dans : European Journal of Medicinal Chemistry. 94, p. 45-55 11 p., 7726

Résultats de recherche: Contribution à un journal/une revueArticle

Accès ouvert
Harmine
Quantitative Structure-Activity Relationship
Solubility
In Vitro Techniques
Derivatives
Harmine
Cyclodextrins
Solubility
Pharmaceutical Preparations
Protons
lead compounds
polymorphism
thiols
solid state
predictions
2013

Indoleamine 2,3-Dioxygenase Inhibitory Activity of Derivatives of Marine Alkaloid Tsitsikammamine A

Dolusic, E., Larrieu, P., Meinguet, C., Colette, D., Rives, A., Blanc, S., Ferain, T., Pilotte, L., Stroobant, V., Wouters, J., Van den Eynde, B., Masereel, B., Delfourne, E. & Frédérick, R. 1 janv. 2013 Dans : Bioorganic and medicinal chemistry letters. 23, 1, p. 47-54 8 p.

Résultats de recherche: Contribution à un journal/une revueArticle

Indoleamine-Pyrrole 2,3,-Dioxygenase
Alkaloids
Assays
Derivatives
tsitsikammamine A
2012

Biochemical and structural characterization of the arabidopsis bifunctional enzyme dethiobiotin synthetase-diaminopelargonic acid aminotransferase: Evidence for substrate channeling in biotin synthesis

Cobessi, D., Meinguet, C., Ferrer, J-L., Dumas, R., Pautre, V. & Alban, C. 1 avr. 2012 Dans : Plant Cell Physiol, . 24, 4, p. 1608-1625 18 p.

Résultats de recherche: Contribution à un journal/une revueArticle

transaminases
biotin
ligases
Arabidopsis
synthesis

Novel trisubstituted harmine derivatives with original in vitro anticancer activity

Frédérick, R., Bruyére, C., Vancraeynest, C., Reniers, J., Meinguet, C., Pochet, L., Backlund, A., Masereel, B., Kiss, R. & Wouters, J. 26 juil. 2012 Dans : Journal of medicinal chemistry. 55, 14, p. 6489-6501 13 p.

Résultats de recherche: Contribution à un journal/une revueArticle

Harmine
Carbolines
Neoplasms
In Vitro Techniques
Growth
2011
Tryptophan Oxygenase
Indoleamine-Pyrrole 2,3,-Dioxygenase
Monoamine Oxidase
Derivatives
Substrates