Résultat de recherche 1989 2017

Filtre
Poster
2013

3-ALKENYL INDOLES AS TRYPTOPHAN 2,3-DIOXYGENASE INHIBITORS FOR THE ENHANCEMENT OF CANCER IMMUNOTHERAPY

Dolušić, E., Pilotte, L., Moineaux, L., Larrieu, P., Stroobant, V., Colau, D., Pochet, L., De Plaen, E., Uyttenhove, C., Van den Eynde, B., Wouters, J., Masereel, B., Lanners, S. & Frédérick, R. 27 mai 2013 p. Book of Abstracts, Heterocycles in Bio-organic Chemistry, Riga, Latvia, 27 - 30 May 2013, PO129 1 p.

Résultats de recherche: Recherche - Revue par des pairsPoster

Accès ouvert
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Tryptophan Oxygenase
Indoles
Tryptophan
Molecular modeling
Tumors
2012

Convenient one-pot formation of highly functionalized 5-halothiazoles

Dolusic, E., Modaffari, S., Pochet, L., Wouters, J., Masereel, B. & Frédérick, R. 1 juil. 2012 p. Book of Abstracts, Balticum Organicum Syntheticum, July 1-4 2012, Tallinn, Estonia, PO27, p. 74 1 p.

Résultats de recherche: RecherchePoster

Accès ouvert
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Thiazoles
Bearings (structural)
Bromine
Oxidants
Oxides

Tryptophan 2,3-Dioxygenase (TDO) Inhibitors as Anticancer Immunomodulators

Dolusic, E., Larrieu, P., Moineaux, L., Strobant, V., Pilotte, L., Colau, D., Pochet, L., De Plaen, E., Uyttenhove, C., Van den Eynde, B., Wouters, J., Masereel, B. & Frédérick, R. 15 juil. 2012 p. Programme & Book of Abstracts, BOSS XIII, KU Leuven, Belgium, 15 - 20 July 2012, P292, p. 339 1 p.

Résultats de recherche: RecherchePoster

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Tryptophan Oxygenase
Immunologic Factors
Tryptophan
Indoleamine-Pyrrole 2,3,-Dioxygenase
Heterocyclic Compounds
2011

A CONVENIENT FORMATION OF HIGHLY FUNCTIONALIZED 5-BROMO-1,3-THIAZOLES.

Dolusic, E., Modaffari, S., Wouters, J., Masereel, B. & Frédérick, R. 2011 p. Book of Abstracts, 15th Sigma-Aldrich Organic Synthesis Meeting, Spa, Belgium, 1-2 December 2011, p. 25 1 p.

Résultats de recherche: RecherchePoster

Accès ouvert
!!File
Thiazoles
Electrons
Bearings (structural)
Bromine
Oxides

Aromatic Thiosemicarazones are inhibitors of tryptophan 2,3-Dioxygenase (TDO), an emerging target for cancer treatment

Dolusic, E., Modaffari, S., Larrieu, P., Vancraeynest, C., Pilotte, L., Colau, D., Stroobant, V., Wouters, J., Masereel, B., Van den Eynde, B. & Frédérick, R. 2011 p. Book of Abstracts, ASMC 11, St. Petersburg, Russia, August 21-25, 2011, P157 1 p.

Résultats de recherche: RecherchePoster

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Tryptophan Oxygenase
Thiosemicarbazones
Oncology
Methisazone
Bearings (structural)

Indole-pyridinyl-ethanones as novel inhibitors of indoleamine-2,3 dioxygenase (IDO), a promising target for anti-cancer immunotherapy

Dolusic, E., Larrieu, P., Blanc, S., Moineaux, L., Sapunaric, F., Pouyez, J., Colette, D., Fraser, G., Stroobant, V., Pilotte, L., Colau, D., Frère, J-M., Masereel, B., Van den Eynde, B., Wouters, J. & Frédérick, R. 2011 p. Book of Abstracts, 47èmes RICT, 6-8 juillet 2011, Lyon, France, IS08, p. 136 1 p.

Résultats de recherche: RecherchePoster

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Indole-pyridinyl-ethanones as novel inhibitors of indoleamine-2,3-dioxygenase (IDO), a promising target for anti-cancer immunotherapy

Dolusic, E., Larrieu, P., Blanc, S., Moineaux, L., Colette, D., Fraser, G., Stroobant, V., Pilotte, L., Colaux, D., Wouters, J., Masereel, B., Van den Eynde, B. & Frédérick, R. 2011 p. Book of Abstracts, 25èmes Journées Franco-belges de Pharmacochimie, 19-20/05/11, Liège, P37, p. 62 1 p.

Résultats de recherche: RecherchePoster

Indoleamine-Pyrrole 2,3,-Dioxygenase
Immunotherapy
Neoplasms
indole
Tryptophan

Novel Inhibitors of Indoleamine 2,3-Dioxygenase (IDO), a Target for Anti-Cancer Immunotherapy

Dolusic, E., Blanc, S., Larrieu, P., Moineaux, L., Colette, D., Fraser, G., Stroobant, V., Pilotte, L., Colau, D., Wouters, J., Masereel, B., Van den Eynde, B. & Frédérick, R. 2011 p. Book of Abstracts, XVIIIème Journée Jeunes Chercheurs, 04/02/11, Paris, France 1 p.

Résultats de recherche: RecherchePoster

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Indoleamine-Pyrrole 2,3,-Dioxygenase
Tryptophan
Tumors
Screening
Cells

SYNTHESIS, ACTIVITY, CRYSTAL AND ELECTRONIC PROPERTIES OF ISOMERS OF CHLORO-PYRIDINYLVINYL-1H-INDOLES

Moineaux, L., Laurent, S., Dolusic, E., Reniers, J., Norberg, B., Frère, J-M., Galleni, M., Van den Eynde, B., Masereel, B., Frédérick, R. & Wouters, J. 2011 p. Book of Abstracts, 25èmes Journées Franco-belges de Pharmacochimie, 19-20/05/11, Liège, P20, p. 45 1 p.

Résultats de recherche: RecherchePoster

Indoles
Tryptophan
Isomers
Electronic properties
Tumors

Synthesis, structural, enzymatic and cellular studies of vinyl-1H-indole analogues as potential inhibitors of tryptophan 2,3-dioxygenase (TDO), an attractive target in cancer immunotherapy.

Moineaux, L., Charlier, C., Dolusic, E., Larrieu, P., Pilotte, L., Colau, D., Stroobant, V., Charlier, P., Laurent, S., Galleni, M., Masereel, B., Van den Eynde, B., Wouters, J. & Frédérick, R. 2011 p. Book of Abstracts, Annual One-Day Meeting on Medicinal Chemistry of SRC & KVCV (MedChem 2011), Ghent, 25 November 2011, p. 22 1 p.

Résultats de recherche: RecherchePoster

THIOSEMICARBAZONES AS INHIBITORS OF TRYPTOPHAN 2,3-DIOXYGENASE (TDO), AN EMERGING TARGET FOR CANCER TREATMENT

Dolusic, E., Modaffari, S., Larrieu, P., Vancraeynest, C., Pilotte, L., Colau, D., Stroobant, V., Van den Eynde, B., Wouters, J., Masereel, B. & Frédérick, R. 2011 p. Book of Abstracts, Annual One-Day Meeting on Medicinal Chemistry of SRC & KVCV (MedChem 2011), Ghent, 25 November 2011, p. 21 1 p.

Résultats de recherche: RecherchePoster

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Tryptophan Oxygenase
Indoleamine-Pyrrole 2,3,-Dioxygenase
Thiosemicarbazones
Oncology
Enzymes

Tryptophan 2,3-dioxygenase (TDO) inhibitors : Identification of new scaffolds using virtual screening

Moineaux, L., Charlier, C., Dolusic, E., Larrieu, P., Pilotte, L., Colau, D., Stroobant, V., Galleni, M., Masereel, B., Van den Eynde, B., Wouters, J. & Frédérick, R. 2011 p. Book of Abstracts, 25èmes Journées Franco-belges de Pharmacochimie, 19-20/05/11, Liège, p. 19 1 p.

Résultats de recherche: RecherchePoster

Accès ouvert
!!File
Tryptophan Oxygenase
Neoplasms
Ralstonia
Posters
Tryptophan
2010

Conception, synthèse et étude d'inhibiteurs de la tryptophane 2,3-dioxygénase (TDO), une cible prometteuse pour le traitement du cancer

Moineaux, L., Charlier, C., Dolusic, E., Larrieu, P., Pilotte, L., Colau, D., Stroobant, V., Galleni, M., Masereel, B., Van den Eynde, B., Wouters, J. & Frédérick, R. 2010 p. Abstracts, Séminaire des jeunes chercheurs Télévie 2011, Brussels, Belgium, 7 December 2010 1 p.

Résultats de recherche: RecherchePoster

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Design, synthesis and study of inhibitors of tryptophan 2,3-dioxygenase (TDO), a promising target for cancer therapy

Moineaux, L., Charlier, C., Dolusic, E., Larrieu, P., Pilotte, L., Colau, D., Stroobant, V., Galleni, M., Masereel, B., Van den Eynde, B., Wouters, J. & Frédérick, R. 2010 p. Abstracts, école doctorale SFMBBM, Liège, Belgium, 10 December 2010 1 p.

Résultats de recherche: RecherchePoster

Tryptophan Oxygenase
Neoplasms
Therapeutics
Tryptophan
Enzymes

Discovery and Optimization Of Indole-pyridinyl-ethanones as Novel Inhibitors of Indoleamine-2,3-Dioxygenase (IDO), a Promising Target for Anti-Cancer Immunotherapy

Frédérick, R., Blanc, S., Larrieu, P., Moineaux, L., Colette, D., Fraser, G., Stroobant, V., Pilotte, L., Colau, D., Wouters, J., Masereel, B., Van den Eynde, B. & Dolusic, E. 2010 p. PC.281, 21st ISMC, Brussels, Belgium, September 5-9, 2010, Drugs of the Future, volume 35, issue suppl. A, pp. 181-182 2 p.

Résultats de recherche: RecherchePoster

Tryptophan Oxygenase
Indoleamine-Pyrrole 2,3,-Dioxygenase
Tumors
indole
Enzyme inhibition

Indole-pyridinyl-ethanones as Novel Inhibitors of Indoleamine 2,3-Dioxygenase (IDO), a Promising Target forAnti-Cancer Immunotherapy

Dolusic, E., Blanc, S., Larrieu, P., Moineaux, L., Colette, D., Fraser, G., Stroobant, V., Pilotte, L., Colau, D., Wouters, J., Masereel, B., Van den Eynde, B. & Frédérick, R. 2010 p. Book of Abstracts, XXIVth European Colloquium on Heterocyclic Chemistry, Vienna, Austria, August 23-27, 2010 1 p.

Résultats de recherche: RecherchePoster

Accès ouvert
!!File
Indoleamine-Pyrrole 2,3,-Dioxygenase
Immunotherapy
Neoplasms
indole
Tryptophan

Synthesis, crystal and electronic properties of isomers of chloro-pyridinylvinyl-1H-indoles

Moineaux, L., Charlier, C., Dolusic, E., Larrieu, P., Pilotte, L., Colau, D., Stroobant, V., Galleni, M., Masereel, B., Van den Eynde, B., Wouters, J. & Frédérick, R. 2010 p. Abstracts, The sixth Belgian Crystallography Symposium (BCS-6), 13 October 2010, Brussels, Belgium 1 p.

Résultats de recherche: RecherchePoster

Indoles
Neoplasms
Enzymes
Tryptophan
Therapeutics

Tryptophan 2,3-dioxygenase (TDO) inhibitors : Identification of new scaffolds using virtual screening

Moineaux, L., Charlier, C., Dolusic, E., Larrieu, P., Pilotte, L., Colau, D., Stroobant, V., Galleni, M., Masereel, B., Van den Eynde, B., Wouters, J. & Frédérick, R. 2010 p. Abstracts, Journée scientifique de la Société royale de chimie (SRC), Gembloux, Belgium, 14 October 2010

Résultats de recherche: RecherchePoster

!!File
Tryptophan Oxygenase
Neoplasms
Tryptophan
Enzymes
Therapeutics
1991

New relative K+-sparing high ceiling diuretics related to torasemide.

Masereel, B., Schynts, M., Lohrmann, E., Pirotte, B. & Delarge, J. 1991

Résultats de recherche: Recherche - Revue par des pairsPoster

1990

New sulfonylurea derivatives as potential antihypertensive drugs.

Masereel, B., Pirotte, B., Schynts, M., Ferrari, P., Thunus, L. & Delarge, J. 1990

Résultats de recherche: Recherche - Revue par des pairsPoster

1989

New torasemide derivatives inhibit brain slices and astrocytes swelling induced by potassium.

Masereel, B., Grisar, T., Delarge, J. & Burette, M. 1989

Résultats de recherche: Recherche - Revue par des pairsPoster