Rational design, synthesis, molecular modeling and evaluation of b-carbolines and 5H-indeno[1,2-c]pyridazin-5-one derivatives as potential MAO and IDO inhibitors

Jérémy Reniers; Johan Wouters; Raphaël Frédérick

Rational design, synthesis, molecular modeling and evaluation of b-carbolines and 5H-indeno[1,2-c]pyridazin-5-one derivatives as potential MAO and IDO inhibitors

Jérémy Reniers, Johan Wouters, Raphaël Frédérick

Research output: Other contribution

Original language	English
Publication status	Published - 2011

1 Literature review

Discovery and optimization of indole-pyridinyl-ethanones as novel inhibitors of indoleamine-2-3 dioxygenase (IDO), a promising target for anti-cancer immunotherapy.
Frédérick, R., Blanc, S., Larrieu, P., Moineaux, L., Colette, D., Fraser, G., Stroobant, V., Pilotte, L., Colaux, D., Wouters, J., Masereel, B., Van den Eynde, B. & Dolušić, E., 2010, In: Drugs of the future. 35, suppl A, p. 181-182
Research output: Contribution to journal › Literature review › peer-review

Rational design, synthesis, molecular modeling and evaluation of β-carboline and 5H-indeno[1,2-c]pyridazin-5-one derivatives as potential MAO and IDO inhibitors
Author: Reniers, J., 4 Oct 2011
Supervisor: Wouters, J. (Supervisor), Frederick, R. (Jury), Michiels, C. (Jury), Vincent, S. (President) & Kiss, R. (External person) (Jury)
Student thesis: Doc types › Doctor of Sciences

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Cite this

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title = "Rational design, synthesis, molecular modeling and evaluation of b-carbolines and 5H-indeno[1,2-c]pyridazin-5-one derivatives as potential MAO and IDO inhibitors",

author = "J{\'e}r{\'e}my Reniers and Johan Wouters and Rapha{\"e}l Fr{\'e}d{\'e}rick",

year = "2011",

language = "English",

type = "Other",

}

Rational design, synthesis, molecular modeling and evaluation of b-carbolines and 5H-indeno[1,2-c]pyridazin-5-one derivatives as potential MAO and IDO inhibitors

Research output

Discovery and optimization of indole-pyridinyl-ethanones as novel inhibitors of indoleamine-2-3 dioxygenase (IDO), a promising target for anti-cancer immunotherapy.

Student Theses

Rational design, synthesis, molecular modeling and evaluation of β-carboline and 5H-indeno[1,2-c]pyridazin-5-one derivatives as potential MAO and IDO inhibitors

Cite this