Discovery and optimization of indole-pyridinyl-ethanones as novel inhibitors of indoleamine-2-3 dioxygenase (IDO), a promising target for anti-cancer immunotherapy.

Raphaël Frédérick; Sébastien Blanc; Pierre Larrieu; Laurence Moineaux; Delphine Colette; Graeme Fraser; Vincent Stroobant; Luc Pilotte; Didier Colaux; Johan Wouters; Bernard Masereel; Benoît Van den Eynde; Eduard Dolušić

Discovery and optimization of indole-pyridinyl-ethanones as novel inhibitors of indoleamine-2-3 dioxygenase (IDO), a promising target for anti-cancer immunotherapy.

Raphaël Frédérick, Sébastien Blanc, Pierre Larrieu, Laurence Moineaux, Delphine Colette, Graeme Fraser, Vincent Stroobant, Luc Pilotte, Didier Colaux, Johan Wouters, Bernard Masereel, Benoît Van den Eynde, Eduard Dolušić

Research output: Contribution to journal › Literature review

Original language	French
Pages (from-to)	181-182
Journal	Drugs of the future
Volume	35
Issue number	suppl A
Publication status	Published - 2010

Cite this

Frédérick, R., Blanc, S., Larrieu, P., Moineaux, L., Colette, D., Fraser, G., ... Dolušić, E. (2010). Discovery and optimization of indole-pyridinyl-ethanones as novel inhibitors of indoleamine-2-3 dioxygenase (IDO), a promising target for anti-cancer immunotherapy. Drugs of the future, 35(suppl A), 181-182.

Frédérick, Raphaël ; Blanc, Sébastien ; Larrieu, Pierre ; Moineaux, Laurence ; Colette, Delphine ; Fraser, Graeme ; Stroobant, Vincent ; Pilotte, Luc ; Colaux, Didier ; Wouters, Johan ; Masereel, Bernard ; Van den Eynde, Benoît ; Dolušić, Eduard. / Discovery and optimization of indole-pyridinyl-ethanones as novel inhibitors of indoleamine-2-3 dioxygenase (IDO), a promising target for anti-cancer immunotherapy. In: Drugs of the future. 2010 ; Vol. 35, No. suppl A. pp. 181-182.

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title = "Discovery and optimization of indole-pyridinyl-ethanones as novel inhibitors of indoleamine-2-3 dioxygenase (IDO), a promising target for anti-cancer immunotherapy.",

author = "Rapha{\"e}l Fr{\'e}d{\'e}rick and S{\'e}bastien Blanc and Pierre Larrieu and Laurence Moineaux and Delphine Colette and Graeme Fraser and Vincent Stroobant and Luc Pilotte and Didier Colaux and Johan Wouters and Bernard Masereel and {Van den Eynde}, Beno{\^i}t and Eduard Dolušić",

year = "2010",

language = "Fran{\cc}ais",

volume = "35",

pages = "181--182",

journal = "Drugs of the future",

issn = "0377-8282",

publisher = "Prous Science",

number = "suppl A",

}

Frédérick, R, Blanc, S, Larrieu, P, Moineaux, L, Colette, D, Fraser, G, Stroobant, V, Pilotte, L, Colaux, D, Wouters, J , Masereel, B, Van den Eynde, B & Dolušić, E 2010, 'Discovery and optimization of indole-pyridinyl-ethanones as novel inhibitors of indoleamine-2-3 dioxygenase (IDO), a promising target for anti-cancer immunotherapy.', Drugs of the future, vol. 35, no. suppl A, pp. 181-182.

Discovery and optimization of indole-pyridinyl-ethanones as novel inhibitors of indoleamine-2-3 dioxygenase (IDO), a promising target for anti-cancer immunotherapy. / Frédérick, Raphaël; Blanc, Sébastien; Larrieu, Pierre; Moineaux, Laurence; Colette, Delphine; Fraser, Graeme; Stroobant, Vincent; Pilotte, Luc; Colaux, Didier; Wouters, Johan ; Masereel, Bernard; Van den Eynde, Benoît; Dolušić, Eduard.

In: Drugs of the future, Vol. 35, No. suppl A, 2010, p. 181-182.

Research output: Contribution to journal › Literature review

TY - JOUR

T1 - Discovery and optimization of indole-pyridinyl-ethanones as novel inhibitors of indoleamine-2-3 dioxygenase (IDO), a promising target for anti-cancer immunotherapy.

AU - Frédérick, Raphaël

AU - Blanc, Sébastien

AU - Larrieu, Pierre

AU - Moineaux, Laurence

AU - Colette, Delphine

AU - Fraser, Graeme

AU - Stroobant, Vincent

AU - Pilotte, Luc

AU - Colaux, Didier

AU - Wouters, Johan

AU - Masereel, Bernard

AU - Van den Eynde, Benoît

AU - Dolušić, Eduard

PY - 2010

Y1 - 2010

M3 - Revue de documentation

VL - 35

SP - 181

EP - 182

JO - Drugs of the future

JF - Drugs of the future

SN - 0377-8282

IS - suppl A

ER -

Research Output

Reversal of tumoral immune resistance by inhibition of tryptophan 2,3-dioxygenase

Research output: Contribution to journal › Article

Rational design, synthesis, molecular modeling and evaluation of b-carbolines and 5H-indeno[1,2-c]pyridazin-5-one derivatives as potential MAO and IDO inhibitors

Research output: Other contribution

Tryptophan 2,3-dioxygenase (TDO) inhibitors. 3-(2-(pyridyl)ethenyl)indoles as potential anticancer immunomodulators

Research output: Contribution to journal › Article