Anti-alcohol abuse drug disulfiram inhibits human PHGDH via disruption of its active tetrameric form through a specific cysteine oxidation

Quentin Spillier, Didier Vertommen, Séverine Ravez, Romain Marteau, Quentin Thémans, Cyril Corbet, Olivier Feron, Johan Wouters, Raphaël Frédérick

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Pharmacology, Toxicology and Pharmaceutical Science