@inproceedings{bda79e498ce348b1a8f3f3a3fcd61827,
title = "A general strategy to synthesize ADP-7-Azido-heptose and ADP-Azido-mannoses and their heptosyltransferase binding properties",
abstract = "The multistep synthesis of a novel ADP-7-azido-7-deoxy-l-glycero-β-d-manno-heptopyranoside 2a and several analogues as heptosyltransferase ligands is described. The synthesis of the key intermediate heptoside-1-β-phosphate 3a involved a β-stereoselective phosphorylation of lactol 4 employing diallyl chlorophosphate as a phosphorylating reagent. Five deprotected nucleotide sugars were generated by this synthetic sequence and evaluated as heptosyltransferase substrates (KM, kcat).",
author = "Marine Lacritick",
note = "Funding Information: The authors thank the Fonds National de la Recherche Scientifique (FNRS, mandate “Charg{\'e} de Recherche” for A.T.), CSC (Ph.D. grant for T.L.), National Natural Science Foundation of China (Grant No: 81703364). Additional thanks to Wesleyan University for support for J.M. Publisher Copyright: {\textcopyright} 2021 American Chemical Society. All rights reserved.",
year = "2021",
month = feb,
day = "23",
doi = "10.1021/acs.orglett.1c00048",
language = "English",
volume = "23",
series = "Organic Letters",
pages = "1638--1642",
booktitle = "A general strategy to synthesize ADP-7-Azido-heptose and ADP-Azido-mannoses and their heptosyltransferase binding properties",
edition = "5",
}