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Research Output

Thiosemicarbazide Derivatives as Novel Indolamine-2,3-dioxygenase (IDO) Inhibitors

Serra, S., Moineaux, L., Vancraeynest, C., Masereel, B., Pochet, L., Wouters, J. & Frédérick, R., 2014, Chemmedchem EFMC-ISMC 2014 Book of Abstracts. p. 280

Research output: Contribution in Book/Catalog/Report/Conference proceedingConference contribution

THIOSEMICARBAZONES AS INHIBITORS OF TRYPTOPHAN 2,3-DIOXYGENASE (TDO), AN EMERGING TARGET FOR CANCER TREATMENT

Dolusic, E., Modaffari, S., Larrieu, P., Vancraeynest, C., Pilotte, L., Colau, D., Stroobant, V., Van den Eynde, B., Wouters, J., Masereel, B. & Frédérick, R., 2011, p. Book of Abstracts, Annual One-Day Meeting on Medicinal Chemistry of SRC & KVCV (MedChem 2011), Ghent, 25 November 2011, p. 21. 1 p.

Research output: Contribution to conferencePoster

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Toward Fractioning of Isomers through Binding-Induced Acceleration of Azobenzene Switching

Vulcano, R., Pengo, P., Velari, S., Wouters, J., De Vita, A., Tecilla, P. & Bonifazi, D., 20 Dec 2017, In : Journal of the American Chemical Society. 139, 50, p. 18271-18280 10 p.

Research output: Contribution to journalArticle

Towards new leads for selective carbonic anhydrase IX inhibition: synthesis, pharmacological evaluation and combined ligand-based and target-based approach

Thiry, A., Ledecq, M., Dogné, J-M., SUPURAB, C. T., Wouters, J. & Masereel, B., 2007, Abstract Book-New Drugs and Drug Candidates : Recent Achievements in Medicinal Chemistry.

Research output: Contribution in Book/Catalog/Report/Conference proceedingConference contribution

Towards new leads for selective cyclooxygenase-2 (COX-2) inhibition

Michaux, C., Rolin, S., de Leval, X., Masereel, B., Durant, F. & Wouters, J., 2001, Abstract Book-XVèmes Journées Franco-Belges de Pharmacochimie. Universitaires, P. & Namur, D. (eds.). p. 84

Research output: Contribution in Book/Catalog/Report/Conference proceedingConference contribution

Towards the understanding of the absorption spectra of NAD(P)H/NAD(P)+ as a common indicator of dehydrogenase enzymatic activity

De Ruyck, J., Famerée, M., Wouters, J., Perpète, E. A., Preat, J. & Jacquemin, D., 14 Dec 2007, In : Chemical Physics Letters. 450, 1-3, p. 119-122 4 p.

Research output: Contribution to journalArticle

trans- and cis-S-C-C-S conformations in 5-(2,2′-dithien-5-yl)-2′-deoxyuridine

Wouters, J., Creuven, I., Norberg, B., Evrard, G., Durant, F., Van Aerschot, A. & Herdewijn, P., 15 Jul 1997, In : Acta crystallographica Section C: Crystal Structure communications. 53, 7, p. 892-895 4 p.

Research output: Contribution to journalArticle

Tryptophan 2,3-dioxygenase (TDO) inhibitors : Identification of new scaffolds using virtual screening

Moineaux, L., Charlier, C., Dolusic, E., Larrieu, P., Pilotte, L., Colau, D., Stroobant, V., Galleni, M., Masereel, B., Van den Eynde, B., Wouters, J. & Frédérick, R., 2010, p. Abstracts, Journée scientifique de la Société royale de chimie (SRC), Gembloux, Belgium, 14 October 2010.

Research output: Contribution to conferencePoster

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Tryptophan 2,3-dioxygenase (TDO) inhibitors : Identification of new scaffolds using virtual screening

Moineaux, L., Charlier, C., Dolusic, E., Larrieu, P., Pilotte, L., Colau, D., Stroobant, V., Galleni, M., Masereel, B., Van den Eynde, B., Wouters, J. & Frédérick, R., 2011, p. Book of Abstracts, 25èmes Journées Franco-belges de Pharmacochimie, 19-20/05/11, Liège, p. 19. 1 p.

Research output: Contribution to conferencePoster

Open Access
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Tryptophan 2,3-dioxygenase (TDO) inhibitors. 3-(2-(pyridyl)ethenyl)indoles as potential anticancer immunomodulators

Dolušić, E., Larrieu, P., Moineaux, L., Stroobant, V., Pilotte, L., Colau, D., Pochet, L., Van Den Eynde, B., Masereel, B., Wouters, J. & Frédérick, R., 11 Aug 2011, In : Journal of Medicinal Chemistry. 54, 15, p. 5320-5334 15 p.

Research output: Contribution to journalArticle

Tryptophan 2,3-Dioxygenase (TDO) Inhibitors as Anticancer Immunomodulators

Dolusic, E., Larrieu, P., Moineaux, L., Strobant, V., Pilotte, L., Colau, D., Pochet, L., De Plaen, E., Uyttenhove, C., Van den Eynde, B., Wouters, J., Masereel, B. & Frédérick, R., 15 Jul 2012, p. Programme & Book of Abstracts, BOSS XIII, KU Leuven, Belgium, 15 - 20 July 2012, P292, p. 339. 1 p.

Research output: Contribution to conferencePoster

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236 Downloads (Pure)

Unprecedented copper(I) bifluoride complexes: Synthesis, characterization and reactivity

Vergote, T., Nahra, F., Welle, A., Mager, N., Riant, O., Leyssens, T., Luhmer, M. & Wouters, J., 16 Jan 2012, In : Chemistry: A European Journal. 18, 3, p. 793-798 6 p.

Research output: Contribution to journalArticle

Use of Theoretical Descriptors to Characterize Cation-π Binding Sites in (Macro)molecules

Wouters, J., 30 Jul 2000, In : Journal of Computational Chemistry. 21, 10, p. 847-855 9 p.

Research output: Contribution to journalArticle

Versatile access to benzhydryl-phenylureas through an unexpected rearrangement during microwave-enhanced synthesis of hydantoins

Muccioli, G. G., Wouters, J., Poupaert, J. H., Norberg, B., Poppitz, W., Scriba, G. K. E. & Lambert, D. M., 2 Oct 2003, In : Organic Letters. 5, 20, p. 3599-3602 4 p.

Research output: Contribution to journalArticle

Versatile Self-Adapting Boronic Acids for H-Bond Recognition: From Discrete to Polymeric Supramolecules

Georgiou, I., Kervyn De Meerendre, S., Rossignon, A., De Leo, F., Wouters, J., Bruylants, G. & Bonifazi, D., 22 Feb 2017, In : Journal of the American Chemical Society. 139, 7, p. 2710-2727 18 p.

Research output: Contribution to journalArticle

Wavpred: a wavelet-based algorithm for the prediction of transmembrane proteins

Fischer, P., Baudoux, G. & Wouters, J., 2003, In : Comm. math. sci.. 1, 1, p. 44-56 13 p.

Research output: Contribution to journalArticle

Xylanase XYL1p from Scytalidium acidophilum: Site-directed mutagenesis and acidophilic adaptation

Balaa, B. A., Brijs, K., Gebruers, K., Vandenhaute, J., Wouters, J. & Housen, I., 1 Dec 2009, In : Bioresource technology. 100, 24, p. 6465-6471 7 p.

Research output: Contribution to journalArticle

Yeast epiarginase regulation, an enzyme-enzyme activity control. Identification of residues of ornithine carbamoyltransferase and arginase responsible for enzyme catalytic and regulatory activities

El Alami, M., Dubois, E., Oudjama, Y., Tricot, C., Wouters, J., Stalon, V. & Messenguy, F., 13 Jun 2003, In : Journal of Biological Chemistry. 278, 24, p. 21550-21558 9 p.

Research output: Contribution to journalArticle

Open Access
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Zavalíaite, (Mn,Fe,Mg)(PO ), a new member of the sarcopside group from the La Empleada pegmatite, San Luis Province, Argentina

Hatert, F., Roda-Robles, E., De Parseval, P. & Wouters, J., 1 Dec 2012, In : Canadian Mineralogist. 50, 6, p. 1445-1452 8 p.

Research output: Contribution to journalArticle